Drug Discovery Research

Suven discovery research is focused on discovering and developing new chemical entities (NCEs), which are best in class central nervous system therapies for the treatment of cognitive disorders, major depressive disorders, sleep disorders, psychiatric disorders, pain and inflammation, gastro-intestinal motility disorders. Research targets includes serotonin 6 receptor, serotonin 4 receptor, histamine 3 receptor, Nicotinic acetylcholine (Alpha4beta2) receptor, muscarinic M1 receptor, muscarinic M4 receptor, multimodal (Dopaminergic and seretonergic receptor) and P2X purinoceptor 7 receptor.

CNS Focused Pipeline

Candidates Non-clinical GLP Tox Clinical Phase (US IND) Indication
I II III
Masupirdine

(SUVN-502)
5-HT6 antagonist

Cognition

(Alzheimer's Disease)

Neuropsychiatric Symptoms

(Dementia of Alzheimers's Type)

Samelisant

(SUVN-G3031)

H3 inverse agonist

Narcolepsy
(Sleep Disorders)
        Cognitive Disorders
Usmarapride

(SUVN-D4010)

5-HT4 Partial agonist

 

        Cognitive Disorders
Ropanicant

(SUVN-911)

Alpha4 Beta2 nAChRs antagonist

        Depressive Disorders
SUVN-I6107

M1PAM

Cognitive Disorders
SUVN-M8036

Serotonin/Dopamine

modulator

Psychiatric Disorders
SUVN-D1044

5-HT4 agonist

Gastroinstestinal Disorders

Research Pipeline

Program Devlopment Stage Indication
M1 PAM* Lead Optimization Gastrointestinal Disorders
P2X7 Antagonist Lead Optimization Pain and Inflammation
5-HT1A Agonist Lead Optimization Treatment Resistant Depression
M4 PAM Hit to Lead Psychosis
Multimodal Hit Optimisation Bipolar Disorders